Discovery of the First Highly Selective 1,4-dihydropyrido[3,4-b]pyrazin-3(2H)-one MKK4 Inhibitor

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Discovery of the First Highly Selective 1,4-dihydropyrido[3,4-b]pyrazin-3(2H)-one MKK4 Inhibitor

Author: Katzengruber, Leon; Sander, Pascal; Zwirner, Stefan; Rasch, Alexander; Eberlein, Eric; Selig, Roland; Albrecht, Wolfgang; Zender, Lars; Laufer, Stefan A.
Tübinger Autor(en):
Katzengruber, Leon
Sander, Pascal
Zwirner, Stefan
Rasch, Alexander
Eberlein, Eric
Selig, Roland
Zender, Lars
Laufer, Stefan
Published in: Journal of Medicinal Chemistry (2025), Bd. 68, H. 14, S. 14782-14805
Verlagsangabe: Washington : Amer Chemical Soc
Language: English
Full text: http://dx.doi.org/10.1021/acs.jmedchem.5c00919
ISSN: 0022-2623
DDC Classifikation: 540 - Chemistry and allied sciences
Dokumentart: Article
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