Linking ATP and allosteric sites to achieve superadditive binding with bivalent EGFR kinase inhibitors

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Linking ATP and allosteric sites to achieve superadditive binding with bivalent EGFR kinase inhibitors

Author: Wittlinger, Florian; Ogboo, Blessing C.; Shevchenko, Ekaterina; Damghani, Tahereh; Pham, Calvin D.; Schaeffner, Ilse K.; Oligny, Brandon T.; Chitnis, Surbhi P.; Beyett, Tyler S.; Rasch, Alexander; Buckley, Brian; Urul, Daniel A.; Shaurova, Tatiana; May, Earl W.; Schaefer, Erik M.; Eck, Michael J.; Hershberger, Pamela A.; Poso, Antti; Laufer, Stefan A.; Heppner, David E.
Tübinger Autor(en):
Wittlinger, Florian
Shevchenko, Ekaterina
Rasch, Alexander
Poso, Antti
Laufer, Stefan
Published in: Communications Chemistry (2024), Bd. 7 (1), Article 38
Verlagsangabe: Berlin : Nature Portfolio
Language: English
Full text: http://dx.doi.org/10.1038/s42004-024-01108-3
ISSN: 2399-3669
DDC Classifikation: 540 - Chemistry and allied sciences
Dokumentart: Article
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