Auflistung nach Autor "Koch, Pierre"

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2-Alkylsulfanyl-4(5)-aryl-5(4)-heteroarylimidazoles: An Overview on Synthetic Strategies and Biological Activity

Koch, Pierre; Ansideri, Francesco (2017)
A Diverse and Versatile Regiospecific Synthesis of Tetrasubstituted Alkylsulfanylimidazoles as p38 Mitogen-Activated Protein Kinase Inhibitors

Ansideri, Francesco; Kuhn, Annette; Koch, Pierre; Andreev, Stanislav; Laufer, Stefan (2018)
A novel LysR-type regulator negatively affects biosynthesis of the immunosuppressant brasilicardin

Stegmann, Evi; Wohlleben, Wolfgang; Buchmann, Anina; Gross, Harald; Eitel, Michael; Koch, Pierre; Schwarz, Paul Niklas (2021)
Addressing a Trapped High-Energy Water: Design and Synthesis of Highly Potent Pyrimidoindole-Based Glycogen Synthase Kinase-3 beta Inhibitors

Andreev, Stanislav; Pantsar, Tatu; Kahlke, Niclas; El-Gokha, Ahmed; Ansideri, Francesco; Geibel, Christian; Koch, Pierre; Laufer, Stefan; Lämmerhofer, Michael (2022)
An optimized and versatile synthesis to pyridinylimidazole-type p38 alpha mitogen activated protein kinase inhibitors

El-Gokha, Ahmed; Laufer, Stefan; Koch, Pierre (2015)
c-Jun N-terminal kinase inhibitors: a patent review (2010-2014)

Gehringer, Matthias; Muth, Felix; Koch, Pierre; Laufer, Stefan (2015)
Design and Synthesis of Highly Selective Brain Penetrant p38 alpha Mitogen-Activated Protein Kinase Inhibitors

Kuhn, Annette; Koch, Pierre; Laufer, Stefan; Tormählen, Niklas M. (2022)
Design, Synthesis and Biological Evaluation of 7-Chloro-9H-pyrimido[4,5-b]indole-based Glycogen Synthase Kinase-3 beta Inhibitors

Pantsar, Tatu; Ansideri, Francesco; Kudolo, Mark; Forster, Michael; Koch, Pierre; Andreev, Stanislav; Laufer, Stefan (2019)
Discovery and Evaluation of Enantiopure 9H-pyrimido[4,5-b]indoles as Nanomolar GSK-3 beta Inhibitors with Improved Metabolic Stability

Andreev, Stanislav; Pantsar, Tatu; El-Gokha, Ahmed; Ansideri, Francesco; Kudolo, Mark; Geibel, Christian; Lämmerhofer, Michael; Laufer, Stefan; Koch, Pierre (2020)
Evaluation of Novel Substituted Furopyridines as Inhibitors of Protein Kinases Related to Tau Pathology in Alzheimer's Disease

Koch, Pierre; Ansideri, Francesco (2021)
Fluorescence polarization-based assays for detecting compounds binding to inactive c-Jun N-terminal kinase 3 and p38 alpha mitogen-activated protein kinase

Ansideri, Francesco; Lange, Andreas; El-Gokha, Ahmed; Böckler, Frank; Koch, Pierre (2016)
Fluorescence polarization-based competition binding assay for c-Jun N-terminal kinases 1 and 2

Ansideri, Francesco; Dammann, Marcel; Koch, Pierre; Böckler, Frank (2017)
From 2-Alkylsulfanylimidazoles to 2-Alkylimidazoles: An Approach towards Metabolically More Stable p38 alpha MAP Kinase Inhibitors

Heider, Fabian Andreas; Haun, Urs; Kudolo, Mark; Sessler, Catharina; Laufer, Stefan; Koch, Pierre; Döring, Eva (2017)
Genetic Engineering in Combination with Semi-Synthesis Leads to a New Route for Gram-Scale Production of the Immunosuppressive Natural Product Brasilicardin A

Eitel, Michael; Buchmann, Anina; Gust, Bertolt; Wohlleben, Wolfgang; Stegmann, Evi; Koch, Pierre; Gross, Harald; Schwarz, Paul Niklas (2021)
Halogen-enriched fragment libraries as chemical probes for harnessing halogen bonding in fragment-based lead discovery

Zimmermann, Markus O.; Lange, Andreas; Wilcken, Rainer; Cieslik, Markus B.; Exner, Thomas Eckart; Koch, Pierre; Böckler, Frank (2014)
Inhibitors of c-Jun N-Terminal Kinases: An Update

Koch, Pierre; Gehringer, Matthias; Laufer, Stefan (2015)
Probing Substituents in the 1-and 3-Position : Tetrahydropyrazino-Annelated Water-Soluble Xanthine Derivatives as Multi-Target Drugs With Potent Adenosine Receptor Antagonistic Activity

Koch, Pierre (2018)
Pyridinylimidazoles as dual glycogen synthase kinase 3 beta/p38 alpha mitogen-activated protein kinase inhibitors

Heider, Fabian Andreas; Ansideri, Francesco; Tesch, Roberta; Pantsar, Tatu; Haun, Urs; Koch, Pierre; Döring, Eva; Laufer, Stefan; Kudolo, Mark (2019)
Pyridinylimidazoles as GSK3 beta Inhibitors: The Impact of Tautomerism on Compound Activity via Water Networks

Heider, Fabian Andreas; Pantsar, Tatu; Kudolo, Mark; Ansideri, Francesco; Laufer, Stefan; Koch, Pierre (2019)
Selective mono-de-O-acetylation of the per-O-acetylated brasilicardin carbohydrate side chain

Eitel, Michael; Gross, Harald; Koch, Pierre; Zinad, Dhafer Saber Khalaf (2021)

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